フォロー
André Horatscheck
André Horatscheck
Senior Investigator, H3D, University Of Cape Town
確認したメール アドレス: uct.ac.za
タイトル
引用先
引用先
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box
J Reader, ME van der Watt, D Taylor, C Le Manach, N Mittal, S Ottilie, ...
Nature communications 12 (1), 269, 2021
672021
Plasmodial kinase inhibitors: license to cure?
DG Cabrera, A Horatscheck, CR Wilson, G Basarab, CJ Eyermann, ...
Journal of Medicinal Chemistry 61 (18), 8061-8077, 2018
542018
Direct experimental evidence for halogen–aryl π interactions in solution from molecular torsion balances
H Sun, A Horatscheck, V Martos, M Bartetzko, U Uhrig, D Lentz, ...
Angewandte Chemie 129 (23), 6554-6558, 2017
352017
Benzoylphosphonate‐Based Photoactive Phosphopeptide Mimetics for Modulation of Protein Tyrosine Phosphatases and Highly Specific Labeling of SH2 Domains
A Horatscheck, S Wagner, J Ortwein, BG Kim, M Lisurek, S Beligny, ...
Angewandte Chemie-International Edition 51 (37), 9441, 2012
302012
Alzheimer’s Disease: Identification and Development of β‐Secretase (BACE‐1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS)
MI Fernández‐Bachiller, A Horatscheck, M Lisurek, J Rademann
ChemMedChem 8 (7), 1041-1056, 2013
182013
Identification and profiling of a novel diazaspiro [3.4] octane chemical series active against multiple stages of the human malaria parasite plasmodium falciparum and …
C Le Manach, J Dam, JG Woodland, G Kaur, LP Khonde, C Brunschwig, ...
Journal of medicinal chemistry 64 (4), 2291-2309, 2021
162021
Identification of 2, 4-disubstituted imidazopyridines as hemozoin formation inhibitors with fast-killing kinetics and in vivo efficacy in the Plasmodium falciparum NSG mouse model
A Horatscheck, A Andrijevic, AT Nchinda, C Le Manach, T Paquet, ...
Journal of medicinal chemistry 63 (21), 13013-13030, 2020
132020
Development of selective inhibitors of phosphatidylinositol 3-kinase C2α
WT Lo, H Belabed, M Kücükdisli, J Metag, Y Roske, P Prokofeva, ...
Nature chemical biology 19 (1), 18-27, 2023
122023
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box. Nat Commun 12: 269
J Reader, ME van der Watt, D Taylor, C Le Manach, N Mittal, S Ottilie, ...
72021
5-Aryl-2-(naphtha-1-yl) sulfonamido-thiazol-4 (5 H)-ones as clathrin inhibitors
MJ Robertson, A Horatscheck, S Sauer, L von Kleist, JR Baker, ...
Organic & Biomolecular Chemistry 14 (47), 11266-11278, 2016
62016
Benzoylphosphonat‐basierte, photoaktive Phosphotyrosinpeptidmimetika zur funktionellen Modulierung von Proteintyrosinphosphatasen und hochspezifischen Markierung von SH2‐Domänen
A Horatscheck, S Wagner, J Ortwein, BG Kim, M Lisurek, S Beligny, ...
Angewandte Chemie-German Edition 124 (37), 9577, 2012
42012
Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition
M Kücükdisli, H Bel-Abed, D Cirillo, WT Lo, NL Efrém, A Horatscheck, ...
Journal of Medicinal Chemistry 66 (20), 14278-14302, 2023
2023
Correction to “Identification of 2, 4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and In Vivo Efficacy in the Plasmodium …
A Horatscheck, A Andrijevic, AT Nchinda, C Le Manach, T Paquet, ...
Journal of Medicinal Chemistry 64 (3), 1762-1762, 2021
2021
Inside Cover: Alzheimer’s Disease: Identification and Development of β‐Secretase (BACE‐1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS)(ChemMedChem 7/2013)
MI Fernández‐Bachiller, A Horatscheck, M Lisurek, J Rademann
ChemMedChem 8 (7), 1022-1022, 2013
2013
Fragment-Based, Photoactive Phosphotyrosine Peptide Mimetics
J Rademann, S Wagner, A Horatscheck
JOURNAL OF PEPTIDE SCIENCE 18, S35-S35, 2012
2012
Benzoylphosphonate als photovernetzbare Phosphotyrosinmimetika
A Horatscheck
2011
M. Lisurek, J. Rademann* 1041–1056 Alzheimer’s Disease: Identification and Development of b-Secretase
MI Fernµndez-Bachiller, A Horatscheck
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論文 1–17