Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box J Reader, ME van der Watt, D Taylor, C Le Manach, N Mittal, S Ottilie, ... Nature communications 12 (1), 269, 2021 | 67 | 2021 |
Plasmodial kinase inhibitors: license to cure? DG Cabrera, A Horatscheck, CR Wilson, G Basarab, CJ Eyermann, ... Journal of Medicinal Chemistry 61 (18), 8061-8077, 2018 | 54 | 2018 |
Direct experimental evidence for halogen–aryl π interactions in solution from molecular torsion balances H Sun, A Horatscheck, V Martos, M Bartetzko, U Uhrig, D Lentz, ... Angewandte Chemie 129 (23), 6554-6558, 2017 | 35 | 2017 |
Benzoylphosphonate‐Based Photoactive Phosphopeptide Mimetics for Modulation of Protein Tyrosine Phosphatases and Highly Specific Labeling of SH2 Domains A Horatscheck, S Wagner, J Ortwein, BG Kim, M Lisurek, S Beligny, ... Angewandte Chemie-International Edition 51 (37), 9441, 2012 | 30 | 2012 |
Alzheimer’s Disease: Identification and Development of β‐Secretase (BACE‐1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS) MI Fernández‐Bachiller, A Horatscheck, M Lisurek, J Rademann ChemMedChem 8 (7), 1041-1056, 2013 | 18 | 2013 |
Identification and profiling of a novel diazaspiro [3.4] octane chemical series active against multiple stages of the human malaria parasite plasmodium falciparum and … C Le Manach, J Dam, JG Woodland, G Kaur, LP Khonde, C Brunschwig, ... Journal of medicinal chemistry 64 (4), 2291-2309, 2021 | 16 | 2021 |
Identification of 2, 4-disubstituted imidazopyridines as hemozoin formation inhibitors with fast-killing kinetics and in vivo efficacy in the Plasmodium falciparum NSG mouse model A Horatscheck, A Andrijevic, AT Nchinda, C Le Manach, T Paquet, ... Journal of medicinal chemistry 63 (21), 13013-13030, 2020 | 13 | 2020 |
Development of selective inhibitors of phosphatidylinositol 3-kinase C2α WT Lo, H Belabed, M Kücükdisli, J Metag, Y Roske, P Prokofeva, ... Nature chemical biology 19 (1), 18-27, 2023 | 12 | 2023 |
Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box. Nat Commun 12: 269 J Reader, ME van der Watt, D Taylor, C Le Manach, N Mittal, S Ottilie, ... | 7 | 2021 |
5-Aryl-2-(naphtha-1-yl) sulfonamido-thiazol-4 (5 H)-ones as clathrin inhibitors MJ Robertson, A Horatscheck, S Sauer, L von Kleist, JR Baker, ... Organic & Biomolecular Chemistry 14 (47), 11266-11278, 2016 | 6 | 2016 |
Benzoylphosphonat‐basierte, photoaktive Phosphotyrosinpeptidmimetika zur funktionellen Modulierung von Proteintyrosinphosphatasen und hochspezifischen Markierung von SH2‐Domänen A Horatscheck, S Wagner, J Ortwein, BG Kim, M Lisurek, S Beligny, ... Angewandte Chemie-German Edition 124 (37), 9577, 2012 | 4 | 2012 |
Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition M Kücükdisli, H Bel-Abed, D Cirillo, WT Lo, NL Efrém, A Horatscheck, ... Journal of Medicinal Chemistry 66 (20), 14278-14302, 2023 | | 2023 |
Correction to “Identification of 2, 4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and In Vivo Efficacy in the Plasmodium … A Horatscheck, A Andrijevic, AT Nchinda, C Le Manach, T Paquet, ... Journal of Medicinal Chemistry 64 (3), 1762-1762, 2021 | | 2021 |
Inside Cover: Alzheimer’s Disease: Identification and Development of β‐Secretase (BACE‐1) Binding Fragments and Inhibitors by Dynamic Ligation Screening (DLS)(ChemMedChem 7/2013) MI Fernández‐Bachiller, A Horatscheck, M Lisurek, J Rademann ChemMedChem 8 (7), 1022-1022, 2013 | | 2013 |
Fragment-Based, Photoactive Phosphotyrosine Peptide Mimetics J Rademann, S Wagner, A Horatscheck JOURNAL OF PEPTIDE SCIENCE 18, S35-S35, 2012 | | 2012 |
Benzoylphosphonate als photovernetzbare Phosphotyrosinmimetika A Horatscheck | | 2011 |
M. Lisurek, J. Rademann* 1041–1056 Alzheimer’s Disease: Identification and Development of b-Secretase MI Fernµndez-Bachiller, A Horatscheck | | |