| Iodine (V) reagents in organic synthesis. Part 1. Synthesis of polycyclic heterocycles via Dess− Martin periodinane-mediated cascade cyclization: generality, scope, and … KC Nicolaou, PS Baran, YL Zhong, K Sugita Journal of the American Chemical Society 124 (10), 2212-2220, 2002 | 176 | 2002 |
| Iodine(V) Reagents in Organic Synthesis. Part 2. Access to Complex Molecular Architectures via Dess−Martin Periodinane-Generated o-Imidoquinones KC Nicolaou, K Sugita, PS Baran, YL Zhong Journal of the American Chemical Society 124 (10), 2221-2232, 2002 | 153 | 2002 |
| Total synthesis of apoptolidin: construction of enantiomerically pure fragments KC Nicolaou, KC Fylaktakidou, H Monenschein, Y Li, B Weyershausen, ... Journal of the American Chemical Society 125 (50), 15433-15442, 2003 | 151 | 2003 |
| Mechanistic Studies of Periodinane‐Mediated Reactions of Anilides and Related Systems KC Nicolaou, PS Baran, R Kranich, YL Zhong, K Sugita, N Zou Angewandte Chemie 113 (1), 208-212, 2001 | 123 | 2001 |
| Total synthesis of apoptolidin: completion of the synthesis and analogue synthesis and evaluation KC Nicolaou, Y Li, K Sugita, H Monenschein, P Guntupalli, HJ Mitchell, ... Journal of the American Chemical Society 125 (50), 15443-15454, 2003 | 120 | 2003 |
| Rheinanthrone, a metabolite of sennoside A, triggers macrophage activation to decrease aquaporin-3 expression in the colon, causing the laxative effect of rhubarb extract R Kon, N Ikarashi, C Nagoya, T Takayama, Y Kusunoki, M Ishii, H Ueda, ... Journal of Ethnopharmacology 152 (1), 190-200, 2014 | 97 | 2014 |
| Angew Chem 113: 213 KC Nicolaou, K Sugita, PS Baran, YL Zhong Angew Chem Int Ed 40, 207, 2001 | 72 | 2001 |
| Total synthesis of apoptolidin: part 2. Coupling of key building blocks and completion of the synthesis KC Nicolaou, Y Li, KC Fylaktakidou, HJ Mitchell, K Sugita Angewandte Chemie International Edition 40 (20), 3854-3857, 2001 | 71 | 2001 |
| Iodoalkyne‐based catalyst‐mediated activation of thioamides through halogen bonding A Matsuzawa, S Takeuchi, K Sugita Chemistry–An Asian Journal 11 (20), 2863-2866, 2016 | 65 | 2016 |
| Structure–activity relationships of bisphenol A analogs at estrogen receptors (ERs): Discovery of an ERα-selective antagonist K Maruyama, M Nakamura, S Tomoshige, K Sugita, M Makishima, ... Bioorganic & medicinal chemistry letters 23 (14), 4031-4036, 2013 | 61 | 2013 |
| Separation of α-glucosidase-inhibitory and liver X receptor-antagonistic activities of phenethylphenyl phthalimide analogs and generation of LXRα-selective antagonists K Motoshima, T Noguchi-Yachide, K Sugita, Y Hashimoto, M Ishikawa Bioorganic & medicinal chemistry 17 (14), 5001-5014, 2009 | 61 | 2009 |
| Anti-influenza activity of phenethylphenylphthalimide analogs derived from thalidomide Y Iwai, H Takahashi, D Hatakeyama, K Motoshima, M Ishikawa, K Sugita, ... Bioorganic & medicinal chemistry 18 (14), 5379-5390, 2010 | 57 | 2010 |
| Activation of Michael acceptors by halogen-bond donors D von der Heiden, E Detmar, R Kuchta, M Breugst Synlett 29 (10), 1307-1313, 2018 | 55 | 2018 |
| Stereocontrolled syntheses of phorbol analogs and evaluation of their binding affinity to PKC K Sugita, CF Neville, M Sodeoka, H Sasai, M Shibasaki Tetrahedron letters 36 (7), 1067-1070, 1995 | 38 | 1995 |
| Mechanistic Studies of Periodinane-Mediated Reaetions of Anilides and Related Systems Stichworter: Anilide. Heterocyclen. Iodreagentien. Oxidationen. Reaktionsmechanismen KC Nicolaou, PS Baran, R Kranich, YL Zhong, K Sugita, N Zou Angewandte Chemie-German Edition 113 (1), 208-212, 2001 | 34 | 2001 |
| Usefulness for the combination of G protein-and β-arrestin-biased ligands of μ-opioid receptors: Prevention of antinociceptive tolerance T Mori, N Kuzumaki, T Arima, M Narita, R Tateishi, T Kondo, Y Hamada, ... Molecular pain 13, 1744806917740030, 2017 | 32 | 2017 |
| Discovery of a new 2-aminobenzhydrol template for highly potent squalene synthase inhibitors M Ichikawa, A Yokomizo, M Itoh, K Sugita, H Usui, H Shimizu, M Suzuki, ... Bioorganic & medicinal chemistry 19 (6), 1930-1949, 2011 | 30 | 2011 |
| Discovery of DF-461, a potent squalene synthase inhibitor M Ichikawa, M Ohtsuka, H Ohki, M Ota, N Haginoya, M Itoh, Y Shibata, ... ACS medicinal chemistry letters 4 (10), 932-936, 2013 | 28 | 2013 |
| Discovery of atrop fixed alkoxy-aminobenzhydrol derivatives: novel, highly potent and orally efficacious squalene synthase inhibitors M Ichikawa, A Yokomizo, M Itoh, N Haginoya, K Sugita, H Usui, ... Bioorganic & medicinal chemistry 19 (17), 5207-5224, 2011 | 28 | 2011 |
| Fused heterocyclic amido compounds as anti-hepatitis C virus agents H Aoyama, K Sugita, M Nakamura, A Aoyama, MTA Salim, M Okamoto, ... Bioorganic & medicinal chemistry 19 (8), 2675-2687, 2011 | 26 | 2011 |
